A Covalent Inhibitor for Glutathione S ‐Transferase Pi (GSTP 1‐1 ) in Human Cells
Abstract
Glutathione S-transferase π (GSTP1-1 ) is overexpressed in many types of cancer and is involved in drug resistance. Therefore, GSTP1-1 is an important target in cancer therapy, and many GST inhibitors have been reported. We had previously developed an irreversible inhibitor, GS-ESF, as an effective GST inhibitor; however, its cellular permeability was too low for it to be used in inhibiting intracellular GST. We have now developed new...
Paper Details
Title
A Covalent Inhibitor for Glutathione S ‐Transferase Pi (GSTP 1‐1 ) in Human Cells
Published Date
Feb 15, 2019
Journal
Volume
20
Issue
7
Pages
900 - 905
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